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Publication

Expansion of chemical space for collaborative lead generation and drug discovery: the European Lead Factory Perspective

Publication
Drug Disc. Today 2015, 20 (11), 1310-1316
Year
2015
Customer
Taros Chemicals
Symeres authors
Jorg Benningshof, Kees Pouwer, Gerhard Müller
Publication

Conformationally restricted k-opioid receptor agonists: Synthesis and pharmacological evaluation of diastereoisomeric and enantiomeric decahydroquinoxalines

Publication
Bioorg. Med. Chem. Lett. 2015, 25 (22), 5326-5330
Year
2015
Customer
Dr. August Wolff
Symeres authors
Peter Molenveld, Renaud Bouzanne des Mazery, Geert Jan Sterk, Roy Storcken, Reshma Autar, Bram van Ossa, Richard van der Haas
Publication

Cyclopentitol as a scaffold for a natural product-like compound library for drug discovery

Publication
Bioorg. Med. Chem. 2015, 23 (11), 2650-2655
Year
2015
Customer
Leinden Institute of Chemicals
Symeres authors
Sjoerd Aertssen, Remco Beuving, Jorg Benningshof
Publication

Separating closely resembling steroids with ionic liquids in liquid–liquid extraction systems

Publication
Separation and Purification Technology 155 (2015) 58–65
Year
2015
Customer
DSM
Symeres authors
Kristel Gibcus, Ton Visser
Publication

Selective recovery of a pyridine derivative from an aqueous waste stream containing acetic acid and succinonitrile with solvent impregnated resins

Publication
Reactive & Functional Polymers 86 (2015) 67–79
Year
2015
Customer
Eindhoven University of Technology
Symeres authors
Ton Visser
Publication

Novel analogs of antitumor agent calixarene 0118: Synthesis, cytotoxicity, click labeling with 2-[18F]fluoroethylazide, and in vivo evaluation

Publication
European Journal of Organic Chemistry 2015, 89, 279–295
Year
2015
Customer
Philips
Symeres authors
Ton Visser
Publication

Novel pantothenate derivatives for anti-malarial chemotherapy

Publication
Malaria Journal (2015), 14, Art.No: 673
Year
2015
Customer
Chiralix
Symeres authors
Richard Blaauw
Publication

Attrition Induced Deracemisation of 2-Fluorophenylglycine

Publication
Org. Process Res. Dev. 2015, 19, 1, 302-308
Year
2014
Customer
RUG
Symeres authors
Maarten van der Meijden, Richard Kellogg
Publication

Van der Waals interactions in the self-assembly of 5-amino[6]helicene on Cu(100) and Au(111)

Publication
Chem. Commun., 2014, 50, 13907
Year
2014
Customer
Centro Atómico Bariloche/ Max Planck
Symeres authors
Maarten van der Meijden, Richard Kellogg
Publication

Localized Crystallization of Enantiomeric Organic Compounds on Chiral Micro-patterns from Various Organic Solutions

Publication
Chem. Eur. J. 2014, 20, 33, 10466–10474
Year
2014
Customer
Symeres authors
Maarten van der Meijden, Richard Kellogg
 
 

Development Centres of Excellence Network Lead Optimization Hit Generation Lead Optimization
 
 
 
 
 

Development Centres of Excellence Network Lead Optimization Hit Generation Lead Optimization
 
 
 
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