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Publication

3-(Arylamino)-1,2,4-triazine-5-one: A Novel Synthesis and its Use

Publication
Eur. J. Org. Chem. 2010, 15, 2852-2854
Year
2010
Customer
Janssen Pharma-ceutica N.V. (CMD)
Site
Nijmegen
Department
Discovery
MCS people
Ruben leenders, Dirk Vandenput, Remco Zijlmans
Publication

6-Phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile as cathepsin S inhibitors

Publication
Bioorg. Med. Chem. Lett. 2010, 20, 4350–4354
Year
2010
Customer
MSD Newhouse
Site
Nijmegen
Department
Discovery
MCS people
Leon van Berkom, Martijn Bastiani, Tommi Meulemans
Publication

Biotransformation-mediated synthesis of (1S)-1-(2,6-dichloro-3-fluorophenyl)ethanol in enantiomerically pure form

Publication
Tetrahedron: Asymmetry 2010, 21, 19, 2408-2412
Year
2010
Customer
Pfizer
Site
Groningen
Department
MCS people
Erik Keller, Renzo Meijer, Gerard Metselaar, Gerlof Kruidhof
Publication

Practical Aspects of Carbon Carbon Cross-Coupling Reactions Using Heteroarenes

Publication
Organic Process Research & Development 2010, 14, 30–47
Year
2010
Customer
DSM
Site
Groningen
Department
MCS people
Vincent Slagt, Richard Kellogg
Publication

The Driving Mechanism Behind Attrition-Enhanced Deracemization

Publication
Angew. Chem. Int. Ed., 2010, 49, 8435-8438
Year
2010
Customer
DSM
Site
Groningen
Department
MCS people
Richard Kellogg
Publication

Scaling Up Attrition-Enhanced Deracemization by Use of An Industrial Bead Mill in a Route to Clopidogrel (Plavix)

Publication
Organic Process Research & Development 2010, 14, 908-911
Year
2010
Customer
DSM
Site
Groningen
Department
MCS people
Maarten van der Meijden, Richard Kellogg
Publication

Enantioselective Symmetry Breaking Directed by the Order of Process Steps

Publication
Angew. Chem. Int. Ed., 2010, 49, 2539-2541
Year
2010
Customer
DSM
Site
Groningen
Department
MCS people
Richard Kellogg
Publication

Efficient Havinga-Kondepudi resolution of conglomerate amino acid derivatives by slow cooling and abrasive grinding

Publication
Cryst. Eng. Comm. 2010, 12, 2051
Year
2010
Customer
DSM
Site
Groningen
Department
MCS people
Michel Leeman, Richard Kellogg
Publication

Attrition-enhanced total resolution leads to homochiral families of amino acid derivatives

Publication
Tetrahedron: Asymmetry, 2010, 21, 1191
Year
2010
Customer
DSM
Site
Groningen
Department
MCS people
Michel Leeman, Jesse de Gooijer, Karin Boer, Karen Zwaagstra, Richard Kellogg
Publication

A facile synthesis of 2,3-azaisoindoline

Publication
Tetrahedron Letters 51 (2010) 5859-5860
Year
2010
Customer
Pfizer
Site
Groningen
Department
MCS people
Michel van den Berg, Kees Pouwer

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